1-[2-(三氟甲基)苯基]-环丙胺盐酸盐合成路线 (共 1 条)
反应条件
1: With titanium(IV) isopropylate in diethyl ether
T=-70 - 20°C;
2: With boron trifluoride in diethyl ether
T=20°C; 2 h;
参考文献
GLENMARK PHARMACEUTICALS S.A.; GHARAT, Laxmikant Atmaram; MUTHUKAMAN, Nagarajan; KHAIRATKAR-JOSHI, Neelima; KATTIGE, Vidya Ganapati
Patent: WO2013/186692 A1, 2013 ;
Location in patent: Page/Page column 69; 70 ;