反应条件
sodium hydrogencarbonate in N,N-dimethyl acetamide
1.) RT, 24 h, 2.) 40 deg C, 2 h;
参考文献
Temple, Carroll; Wheeler, Glynn P.; Elliott, Robert D.; Rose, Jerry D.; Kussner, Conrad L.; et al.
Journal of Medicinal Chemistry, 1982 , vol. 25, # 9 p. 1045 - 1050