2-甲基-2-丙基4-{[(2-溴苄基)氨基]甲基}-1-哌啶羧酸酯合成路线 (共 1 条)
反应条件
sodium tris(acetoxy)borohydride in 1,2-dichloro-ethane
T=20°C; 3 h;
参考文献
Budzik, Brian; Garzya, Vincenzo; Shi, Dongchuan; Walker, Graham; Lauchart, Yann; Lucas, Adam J.; Rivero, Ralph A.; Langmead, Christopher J.; Watson, Jeannette; Wu, Zining; Forbes, Ian T.; Jin, Jian
Bioorganic and Medicinal Chemistry Letters, 2010 , vol. 20, # 12 p. 3545 - 3549