1-[5-(4-氟苯基)-1,2-恶唑-3-基]乙酮合成路线 (共 1 条)
反应条件
triethylamine in tetrahydrofuran; toluene
T=5 - 10°C; 2 h;
参考文献
GILEAD PHARMASSET, LLC; SOFIA, Michael, Joseph; KAKARLA, Ramesh; LIU, Jian; NADUTHAMBI, Devan; MOSLEY, Ralph; STEUER, Holly, Micolochick
Patent: WO2012/103113 A1, 2012 ;
Location in patent: Page/Page column 430-431 ;