反应条件
sodium hydride
1.) DMF, 20 deg C, 30 min, 2.) DMF, 60 deg C, 5 d; Yield given. Multistep reaction;
参考文献
Blackburn, Thomas P.; Cox, Barry; Guildford, Allen J.; Count, David J. Le; Middlemiss, Derek N.; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 12 p. 2252 - 2259