反应条件
1: 68 percent / POCl3 / 4 h / 140 - 150 °C / in sealed tube
2: 10 percent / pyridine / 65-70 deg C, 40 min, then reflux, 2 h
View Scheme
参考文献
Pochat, Francis; Lavelle, Francois; Fizames, Christian; Zerial, Aurelio
European Journal of Medicinal Chemistry, 1987 , vol. 22, p. 135 - 138