反应条件
1: POCl3 / Heating
2: 1) NH3 (liquid), 2) NaOH / 1) 90 to 100 deg C, 12 h, 2) EtOH, water, 45 to 50 deg C, 10 h
View Scheme
参考文献
Bare; McLaren; Campbell; Firor; Resch; Walters; Salama; Meiners; Patel
Journal of Medicinal Chemistry, 1989 , vol. 32, # 12 p. 2561 - 2573