反应条件
1: 73 percent / pyridine, p-toluenesulfonyl chloride / dimethylformamide / 4 h / Heating
2: 40 percent / NaN3, NH4Cl / dimethylformamide / 90 h / Heating
View Scheme
参考文献
Unangst; Carethers; Webster; Janik; Robichaud
Journal of Medicinal Chemistry, 1984 , vol. 27, # 12 p. 1629 - 1633
