反应条件
1: 1.)NH2OH*HCl, MeONa
2: 80 percent / NaH / xylene
3: 1.)Me3SiI, 2.)H2O / or hydrogenolysis over 10percent Pd/C
View Scheme
参考文献
Nikishin, Gennady I.; Troyansky, Emmanuil I.; Svitanko, Igor V.; Chizhov, Oleg S.
Tetrahedron Letters, 1984 , vol. 25, # 1 p. 97 - 98