反应条件
1: 47 percent / CuCl, N-ethylmorpholine / various solvent(s) / 4 h / 140 °C
2: diethyl phosphorocyanidate / dimethylformamide / 0.5 h / 90 °C
3: HOAc, H2SO4 / 1 h / Heating
View Scheme
参考文献
Atwell, Graham J.; Rewcastle, Gordon W.; Baguley, Bruce C.; Denny, William A.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 4 p. 664 - 669
