5-溴-2-氯-4-(4-氟苯基)-6-异丙基嘧啶合成路线 (共 1 条)
反应条件
1: With trichlorophosphate
T=90°C; 2.5 h;
2: With sodium hydrogencarbonate in water; ethyl acetate
Neutrality;
参考文献
ASTRAZENECA UK LIMITED
Patent: WO2007/7119 A1, 2007 ;
Location in patent: Page/Page column 6; 23 ;
WO 2007/007119 A1