反应条件
1: 4-amino-1H-pyrazole-3-carboxylic acid methyl ester With sodium hydroxide in 1,4-dioxane; water
T=15 - 55°C; 5 h;
2: di-tert-butyl dicarbonate in 1,4-dioxane; water
T=50 - 55°C; 2 - 19 h;
3: With hydrogenchloride in water
pH=2; Product distribution / selectivity;