2,5-二氯-4-(三氟甲基)吡啶合成路线 (共 1 条)
反应条件
1: (trifluoromethyl)-trimethylsilane With N-methyl-pyrrolidine; potassium fluoride; copper(l) iodide T=50°C; 1.16667 h; Heating / reflux; 2: 2,5-dichloro-4-iodo-pyridine 20 h; 3: With ammonia; water
参考文献
WO2009/66786 A1, ;
Page/Page column 120-121 ;