2-乙酰氨基-6-氯-吡啶并[3,2-d]嘧啶-4(3h)-酮合成路线 (共 2 条)
反应条件
2 h; Heating / reflux;
参考文献
4 AZA Bioscience nv
Patent: WO2006/135993 A1, 2006 ;
Location in patent: Page/Page column 91-92 ;
反应条件
N-ethyl-N,N-diisopropylamine; trichlorophosphate in 1,4-dioxane
T=20°C; 2 h;
参考文献
4 AZA Bioscience nv
Patent: WO2006/135993 A1, 2006 ;
Location in patent: Page/Page column 95; 100 ;