triethylamine; trichlorophosphate in dichloromethane
参考文献
Vig, O. P.; Trehan, I. R.; Kad, G. L.; Dhawan, R. K.; Grewal, M. S.
Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1980 , vol. 19, # 8 p. 688 - 691
1: 2-methoxy-phenylamine With hydrogenchloride; sodium nitrite in water
Cooling;
2: 1H-benzo[d]imidazole With sodium acetate in water
T=20°C; 51 h; Cooling;
参考文献
Sharma, Deepika; Narasimhan, Balasubramanian; Kumar, Pradeep; Jalbout, Abraham
European Journal of Medicinal Chemistry, 2009 , vol. 44, # 3 p. 1119 - 1127
1: durch Sulfurieren
2: Nitrierung mit Salpeterschwefelsaeure, Hydrolyse, Reduktion der Nitrogruppe und Behandlung mit Acetanhydrid in waessr. Loesung
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