Tsang, W. C. Peter; Munday, Rachel H.; Brasche, Gordon; Zheng, Nan; Buchwald, Stephen L.
Journal of Organic Chemistry, 2008 , vol. 73, # 19 p. 7603 - 7610
1: With acetic acid; sodium nitrite in water
T=0°C; 1 h; Cooling with iceInert atmosphere;
2: With sodium azide in water
T=0 - 20°C; Inert atmosphere;
参考文献
Stokes, Benjamin J.; Jovanovic, Brankica; Dong, Huijun; Richert, Kathleen J.; Riell, Ryan D.; Driver, Tom G.
Journal of Organic Chemistry, 2009 , vol. 74, # 8 p. 3225 - 3228