1: With water; bis-[(trifluoroacetoxy)iodo]benzene in acetonitrile T=65°C; 30 h; 2: With hydrogenchloride in water; acetonitrile pH=1; 3: With sodium carbonate in water pH=8 - 9;
参考文献
NOVARTIS AG; NOVARTIS PHARMA GMBH
Patent: WO2007/121923 A1, 2007 ;
Location in patent: Page/Page column 88 ;
WO 2007/121923 A1