1: 73 percent / Jones' reagent / acetone
2: 90 percent / methanol; K2CO3; water / 2 h / 20 °C
3: 86 percent / acetyl chloride / 24 h / 20 °C
4: phosphate buffer; α-chymotrypsin; sodium hydroxide / 18 h / pH 7.5 / Enzymatic reaction
View Scheme
参考文献
Kim, Dong H.; Park, Jeong-il; Chung, Sang J.; Park, Jung Dae; Park, No-Kyung; Han, Jong Hoon
Bioorganic and Medicinal Chemistry, 2002 , vol. 10, # 8 p. 2553 - 2560