3-溴-5,6,7,8-四氢-[1,2,4]三唑并[4,3-A]吡嗪盐酸盐合成路线 (共 1 条)
反应条件
trifluoroacetic acid in dichloromethane T=0 - 20°C; 16 h;
参考文献
CANCER RESEARCH TECHNOLOGY LIMITED; HOELDER, Swen; BLAGG, Julian; CHEUNG, Jack; ATRASH, Butrus; SHELDRAKE, Peter
Patent: WO2014/37751 A1, 2014 ;
Location in patent: Paragraph 00459-00461 ;