反应条件
1: N,N-dimethyl-2-methylimidazole-1-sulphonamide With n-butyllithium in tetrahydrofuran; hexane T=-78°C; 0.5 h; 2: N,N-dimethyl-formamide in tetrahydrofuran; hexane T=-78 - 20°C; Further stages.;
参考文献
Madsen, Christian; Jensen, Anders A.; Liljefors, Tommy; Kristiansen, Uffe; Nielsen, Birgitte; Hansen, Camilla P.; Larsen, Mogens; Ebert, Bjarke; Bang-Andersen, Benny; Krogsgaard-Larsen, Povl; Frolund, Bente
Journal of Medicinal Chemistry, 2007 , vol. 50, # 17 p. 4147 - 4161