2-甲基氨基嘧啶-5-硼酸频那醇酯合成路线 (共 1 条)
反应条件
potassium acetate; dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct in N,N-dimethyl-formamide
T=80°C; 2 h; Inert atmosphere;
参考文献
DAIICHI SANKYO COMPANY, LIMITED
Patent: US2010/130492 A1, 2010 ;
Location in patent: Page/Page column 93 ;