反应条件
1: sodium hydroxide / water; tetrahydrofuran / 16 h / 0 - 26 °C
2: potassium carbonate / N,N-dimethyl-formamide / 18 h / 22 - 26 °C
3: dihydrogen peroxide / water; ethyl acetate / 2 h / 22 - 26 °C
View Scheme
参考文献
GLENMARK PHARMACEUTICALS S.A.; GHARAT, Laxmikant Atmaram; BANERJEE, Abhisek; PAWAR, Mahesh Yashwant; KHAIRATKAR-JOSHI, Neelima; KATTIGE, Vidya Ganapati
Patent: WO2013/38308 A1, 2013 ;