反应条件
1.1: N,O-bis-(trimethylsilyl)-acetamide / acetonitrile / 80 °C / |Inert atmosphere; |Sealed tube 1.2: 1.08 h / 0 - 80 °C / |Inert atmosphere; |Sealed tube 2.1: ammonia / methanol / 24 h / 20 °C / |Sealed tube View Scheme
参考文献
Vodnala, Suman K.; Lundbaeck, Thomas; Yeheskieli, Esther; Sjoeberg, Birger; Gustavsson, Anna-Lena; Svensson, Richard; Olivera, Gabriela C.; Eze, Anthonius A.; De Koning, Harry P.; Hammarstroem, Lars G. J.; Rottenberg, Martin E.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 24 p. 9861 - 9873
