(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚合成路线

参考文献

Fraley, Mark E.; Arrington, Kenneth L.; Buser, Carolyn A.; Ciecko, Patrice A.; Coll, Kathleen E.; Fernandes, Christine; Hartman, George D.; Hoffman, William F.; Lynch, Joseph J.; McFall, Rosemary C.; Rickert, Keith; Singh, Romi; Smith, Sheri; Thomas, Kenneth A.; Wong, Bradley K.
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 2 p. 351 - 355

7790-94-5氯磺酸+

90732-28-8(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚

210691-38-61-(2,2,2-三氟乙酰基)吲哚啉-5-磺酰氯

参考文献

ANACOR PHARMACEUTICALS, INC.; HERNANDEZ, Vincent, S.; LI, Xianfeng; ZHANG, Suoming; AKAMA, Tsutomu; ZHANG, Yanchen; LIU, Yang; PLATTNER, Jacob, J.; ALLEY, Michael, Kevin Richard; ZHOU, Yasheen; NEIMAN, James, A.
Patent: WO2011/60196 A1, 2011 ;
Location in patent: Page/Page column 129 ;

90732-28-8(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚+

75-36-5乙酰氯

16078-34-51-(2,3-二氢-1H-吲哚-5-基)-乙酮+

147265-76-71-(2,3-二氢-1H-吲哚-6-基)乙酮

参考文献

Ishihara, Yuji; Tanaka, Toshimasa; Goto, Giichi
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1992 , # 24 p. 3401 - 3406

496-15-1吲哚啉+

383-63-1三氟乙酸乙酯

90732-28-8(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚

参考文献

Wyeth
Patent: US2009/48282 A1, 2009 ;
Location in patent: Page/Page column 17 ;

496-15-1吲哚啉+

407-25-0三氟乙酸酐

90732-28-8(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚

参考文献

Fraley, Mark E.; Arrington, Kenneth L.; Buser, Carolyn A.; Ciecko, Patrice A.; Coll, Kathleen E.; Fernandes, Christine; Hartman, George D.; Hoffman, William F.; Lynch, Joseph J.; McFall, Rosemary C.; Rickert, Keith; Singh, Romi; Smith, Sheri; Thomas, Kenneth A.; Wong, Bradley K.
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 2 p. 351 - 355

90732-28-8(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚

参考文献

UNIVERSITY OF SOUTH FLORIDA; WU, Jie; LAWRENCE, Nicholas, J.; SEBTI, Said, M.
Patent: WO2010/11666 A2, 2010 ;
Location in patent: Page/Page column 55-56 ;

5339-85-52-氨基苯乙醇+

76-05-1三氟乙酸

90732-28-8(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚

参考文献

Wang, Zengxue; Wan, Wen; Jiang, Haizhen; Hao, Jian
Journal of Organic Chemistry, 2007 , vol. 72, # 24 p. 9364 - 9367

5339-85-52-氨基苯乙醇+

76-05-1三氟乙酸

参考文献

Wang, Zengxue; Wan, Wen; Jiang, Haizhen; Hao, Jian
Journal of Organic Chemistry, 2007 , vol. 72, # 24 p. 9364 - 9367

120-72-9吲哚

90732-28-8(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚

参考文献

Gribble, Gordon W.; Nutaitis, Charles F.; Leese, Robert M.
Heterocycles, 1984 , vol. 22, # 2 p. 379 - 386

90732-28-8(9ci)-2,3-二氢-1-(三氟乙酰基)-1H-吲哚

823786-82-9

参考文献

Kim, Semi; Park, Ji Hyun; Koo, Sun-Young; Kim, Jung In; Kim, Min-Hyeung; Kim, Ji Eun; Jo, Kiwon; Geun Choi, Hwan; Lee, Sung Bae; Jung, Sang-Hun
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 24 p. 6075 - 6078