反应条件
1.1: sodium hydride / mineral oil; N,N-dimethyl-formamide / 0 °C / |Inert atmosphere
1.2: 20 °C
2.1: hydrogen; palladium 10 on activated carbon / tetrahydrofuran / 20 °C / 2585.81 Torr / |Inert atmosphere
View Scheme
参考文献
THE UNIVERSITY OF NOTTINGHAM; MISTRY, Shailesh; DARAS, Etienne; FROMONT, Christophe; JADHAV, Gopal; FISCHER, Peter Martin; KELLAM, Barrie; HILL, Stephen John; BAKER, Jillian Glenda
Patent: WO2013/121209 A1, 2013 ;