7-氟-6-硝基-1,2,3,4-四氢异喹啉盐酸盐合成路线 (共 2 条)
反应条件
hydrogenchloride; methanol; water
11 h; Heating / reflux;
参考文献
GLAXO GROUP LIMITED
Patent: WO2006/108709 A1, 2006 ;
Location in patent: Page/Page column 51 ;
WO 2006/108709 A1
反应条件
triethylamine in 1,4-dioxane; water
T=20°C; 22 h;
参考文献
GLAXO GROUP LIMITED
Patent: WO2006/108709 A1, 2006 ;
Location in patent: Page/Page column 51 ;
WO 2006/108709 A1