反应条件
1: 92 percent / p-toluenesulfonic acid monohydrate / methanol / Heating
2: 1.) NEt3; 2.) KCl (0.1N) / 1.) CHCl3, room temp., 6h; 40 deg C, 12 h; 2.) 1 h
View Scheme
参考文献
Ohno; Fujita; Nakai; Kobayashi; Inoue; Nojima
Chemical and Pharmaceutical Bulletin, 1985 , vol. 33, # 2 p. 572 - 582