1: With lithium diisopropyl amide in tetrahydrofuran; n-heptane; ethylbenzene
T=0°C; 3 h;
2: With hydrogenchloride; water in tetrahydrofuran; n-heptane; ethylbenzene
T=20°C; 1 h;
参考文献
Kyowa Hakko Kirin Co., Ltd.
Patent: EP2108642 A1, 2009 ;
Location in patent: Page/Page column 87 ;