1: acetyl chloride With AlCl3, aluminium chloride in dichloromethane
T=-7 - 20°C; 0.5 h;
2: 3-phenylpropionyl chloride in dichloromethane
T=0°C;
3: With hydrogenchloride in dichloromethane; water
T=10°C; 1.5 h;
参考文献
SANOFI; BAILLY, Frederic; BON, Xavier; VAYRON, Philippe
Patent: US2013/165674 A1, 2013 ;
Location in patent: Paragraph 0151-0155 ;