1-[(4-碘苯基)磺酰基]-4-甲基哌嗪合成路线 (共 2 条)
反应条件
in tetrahydrofuran
T=20°C;
参考文献
AMGEN INC.
Patent: WO2006/4658 A2, 2006 ;
Location in patent: Page/Page column 52 ;
WO 2006/004658 A2
反应条件
potassium acetate; palladium diacetate in N,N-dimethyl-formamide
T=85°C; 2.5 h;
参考文献
Desos, Patrice; Cordi, Alexis; Lestage, Pierre
Patent: US2006/258670 A1, 2006 ;
Location in patent: Page/Page column 6 ;