1H-吲唑-7-硼酸频哪醇酯合成路线 （共 4 条）
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in dimethyl sulfoxide T=100°C; 48 h;
参考文献
LOCUS PHARMACEUTICALS, INC.
Patent: WO2008/8059 A1, 2008 ;
Location in patent: Page/Page column 66 ;
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in dimethyl sulfoxide T=80°C; 4 h; Product distribution / selectivity;
参考文献
WO2006/46031 A1, ;
Page/Page column 33-35 ;
WO 2006/046031 A1
反应条件
2-(1H-indazol-4-yl)-6-((3R,5S)-3,5-dimethyl-4-thiazol-2-ylmethyl-piperazin-1-ylmethyl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidine in methanol 5 h; Product distribution / selectivity;
参考文献
WO2006/46031 A1, ;
Page/Page column 31-33 ;
WO 2006/046031 A1
反应条件
hydrogenchloride in water T=80°C; 20 h;
参考文献
LOCUS PHARMACEUTICALS, INC.
Patent: WO2008/8059 A1, 2008 ;
Location in patent: Page/Page column 65; 66 ;
