4-溴-5-氯-1-[(4-甲基苯基)磺酰基]-1H-吡咯[2,3-B]吡啶合成路线 (共 1 条)
反应条件
sodium hydride in N,N-dimethyl-formamide
T=0 - 20°C; 2 h;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED
Patent: WO2006/127587 A1, 2006 ;
Location in patent: Page/Page column 87-88 ;
WO 2006/127587 A1