1: With AlCl3, aluminium chloride
Friedel Crafts Arylation;
2: With sodium hydroxide; water
pH=~ 14;
参考文献
ASTEX THERAPEUTICS LIMITED; THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL; CANCER RESEARCH TECHNOLOGY LIMITED; ASTRAZENECA AB
Patent: WO2006/136830 A1, 2006 ;
Location in patent: Page/Page column 193-194 ;
WO 2006/136830 A1