N,N-二甲基-5-碘-1H-吡唑-1-磺酰胺合成路线 (共 1 条)
反应条件
potassium phosphate; palladium diacetate; tri-cyclo-hexyl-phosphine in water; toluene
T=100°C; 2 h;
参考文献
ASTEX THERAPEUTICS LIMITED; THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL; CANCER RESEARCH TECHNOLOGY LIMITED; ASTRAZENECA AB
Patent: WO2006/136830 A1, 2006 ;
Location in patent: Page/Page column 204-205 ;
WO 2006/136830 A1