反应条件
1: oxalyl chloride / N,N-dimethylformamide / CH2Cl2
2: 3.05 g / N-ethyl-N,N-diisopropylamine / CH2Cl2
View Scheme
参考文献
Elsinghorst, Paul W.; Gonzalez Tanarro, Camino M.; Guetschow, Michael
Journal of Medicinal Chemistry, 2006 , vol. 49, # 25 p. 7540 - 7544