1: With sodium bis(2-methoxyethoxy)aluminium dihydride in tetrahydrofuran; toluene T=0 - 20°C; 17 h; 2: With potassium hydroxide; water in tetrahydrofuran; toluene T=0°C;
参考文献
CANCER RESEARCH TECHNOLOGY LIMITED
Patent: WO2009/44162 A1, 2009 ;
Location in patent: Page/Page column 263 ;
WO 2009/044162 A1