反应条件
1: N-benzyl-3-(trimethylsilyloxy)azetidine With hydrogen; palladium dihydroxide in methanol
2: 1,2,3-trifluoro-5-nitrobenzene With N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide
T=45°C; Further stages.;
参考文献
Renslo, Adam R.; Atuegbu, Andy; Herradura, Prudencio; Jaishankar, Priyadarshini; Ji, Mingzhe; Leach, Karen L.; Huband, Michael D.; Dermyer, Michael R.; Wu, Luping; Vara Prasad; Gordeev, Mikhail F.
Bioorganic and Medicinal Chemistry Letters, 2007 , vol. 17, # 18 p. 5036 - 5040
