4-[[5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-3-吡啶]甲基]-吗啉合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane
T=85°C; 8 h; Inert atmosphere;
参考文献
PROGENICS PHARMACEUTICALS, INC.
Patent: WO2009/155527 A2, 2009 ;
Location in patent: Page/Page column 136 ;
WO 2009/155527 A2