4-氯-1H-吡咯并[2,3-B]吡啶-5-羧酸苯甲酯合成路线 (共 1 条)
反应条件
4-(N,N-dimethlyamino)pyridine; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride in N,N-dimethyl-formamide
T=20°C; 72 h;
参考文献
ASTELLAS PHARMA INC.
Patent: WO2007/7919 A2, 2007 ;
Location in patent: Page/Page column 62-63 ;
WO 2007/007919 A2