反应条件
chloroformic acid ethyl ester; triethylamine
1.) CH2Cl2, 0 deg C, 45 min, 2.) CH2Cl2, RT, 2 h; Yield given. Multistep reaction;
参考文献
Mach; Leudtke; Unsworth; Boundy; Nowak; Scripko; Elder; Jackson; Hoffman; Evora; Rao; Molinoff; Childers; Ehrenkaufer
Journal of Medicinal Chemistry, 1993 , vol. 36, # 23 p. 3707 - 3720