反应条件
N,N,N',N',N'',N''-hexamethylphosphoric triamide; copper(l) iodide; ethylamine
1.) THF, from -50 deg C to -40 deg C, 2 h, 2.) from -40 deg C to RT, 1 h; Multistep reaction;
参考文献
Lepoittevin; Benezra
Journal of Medicinal Chemistry, 1986 , vol. 29, # 2 p. 287 - 291