1: p-aminobenzonitrile With hydrogenchloride; chloranil in ethanol; water
T=75°C; 0.0333333 - 0.0833333 h;
2: methyl vinyl ketone in ethanol; water
0.5 h;
参考文献
ELI LILLY AND COMPANY
Patent: WO2007/18818 A1, 2007 ;
Location in patent: Page/Page column 10 ;
WO 2007/018818 A1