反应条件
1: 1.) tetrakis(triphenylphosphine)palladium(0) / 1.) THF, RT, 15 min, 2.) THF, diglyme, 120 deg C, 12 h
2: ammonia / methanol / 12 h / 25 °C
View Scheme
参考文献
Chang, George; Mertes, Mathias P.
Tetrahedron Letters, 1984 , vol. 25, # 23 p. 2431 - 2434