反应条件
Stage #1: <a href="#" onclick="return RXDsubstances(event, this, '5434466', constants.ctx, '0')">benzyl tert-butyl malonate</a> <b>With</b> <a href="#" onclick="return RXDsubstances(event, this, '4122952', constants.ctx, '0')">sodium hydride</a> <b>in</b> <a href="#" onclick="return RXDsubstances(event, this, '102391', constants.ctx, '0')">tetrahydrofuran</a> <br />T=0 - 20°C; 0.75 h; <br />Stage #2: <a href="#" onclick="return RXDsubstances(event, this, '969135', constants.ctx, '0')">methyl iodide</a> <b>in</b> <a href="#" onclick="return RXDsubstances(event, this, '102391', constants.ctx, '0')">tetrahydrofuran</a> <br />T=0 - 20°C; <br />
参考文献
DAIICHI PHARMACEUTICAL CO., LTD. Patent: WO2007/20936 A1, 2007 ; Location in patent: Page/Page column 80 ;