(3S)-2-羟基-3-[[(苄氧基)羰基]氨基]己酸甲酯合成路线 (共 2 条)
反应条件
in methanol T=70°C; 48 h;
参考文献
WO2013/136265 A1, ;
Page/Page column 28-29 ;
反应条件
Multi-step reaction with 2 steps 1: methanol / 48 h / 70 °C2: 5 palladium on charcoal; hydrogen / methanol / 48 h
参考文献
DIPHARMA FRANCIS S.R.L.; ATTOLINO, Emanuele; BOVE, Alessio; BRUNOLDI, Enrico; ALLEGRINI, Pietro Patent: WO2013/136265 A1, 2013 ;