5-苄氧基-2,3-二氢-1H-吲哚合成路线 (共 3 条)
反应条件
hydrogenchloride; sodium nitrite
参考文献
Audouin, Corinne; Mestdagh, Nathalie; Lassoie, Marie-Agnes; Houssin, Raymond; Henichart, Jean-Pierre
Bioorganic and Medicinal Chemistry Letters, 2001 , vol. 11, # 6 p. 845 - 848
反应条件
1: tetrahydrofuran / 20 °C 2: 90 percent / H2 / 10percent Pd/C / ethanol / 760.05 Torr View Scheme
参考文献
Stark, Lucy M.; Lin, Xiao-Fa; Flippin, Lee A.
Journal of Organic Chemistry, 2000 , vol. 65, # 10 p. 3227 - 3230
反应条件
1: With sodium cyanoborohydride; acetic acid
T=0°C; 2 h;
2: With sodium hydroxide; water
参考文献
Wyeth
Patent: US2007/72897 A1, 2007 ;
Location in patent: Page/Page column 40 ;