反应条件
1: (PhO)2POCl, Et3N / dioxane
2: NH3 / CHCl3 / 3 h / 20 °C
3: C5H5N / 3 h / 20 °C
4: hydrazine, C5H5N / acetic acid / 0.05 h / 20 °C
View Scheme
参考文献
Marel, G. A. van der; Wille, G.; Westerink, H.; Wang, A. H.-J.; Rich, A.; et al.
Recueil: Journal of the Royal Netherlands Chemical Society, 1982 , vol. 101, # 2 p. 77 - 78