8-溴-6-氯咪唑并[1,2-b]哒嗪盐酸盐合成路线 (共 2 条)
参考文献
KALYPSYS, INC.; KAHRAMAN, Mehmet; SMITH, Nicholas, D.; BONNEFOUS, Celine; NOBLE, Stewart, A.; PAYNE, Joseph, E.
Patent: WO2010/88518 A2, 2010 ;
Location in patent: Page/Page column 91 ;
WO 2010/088518 A2
反应条件
N-bromosuccinmide in chloroform
T=80°C; 1 h;
参考文献
Bristol-Myers Squibb Company
Patent: US2007/78136 A1, 2007 ;
Location in patent: Page/Page column 66 ;
US 20070078136 A1