5-溴-2-(1-吡咯烷)噻唑合成路线 (共 1 条)
反应条件
N-ethyl-N,N-diisopropylamine in tetrahydrofuran
T=120°C; 0.25 h; Microwave irradiation;
参考文献
GLAXO WELLCOME MANUFACTURING PTE LTD; CHEN, Deborah, W.; DUNCAN, Sarah; KING, Nigel, Paul; LEE, Kiew, Ching; MAK, Sing, Yeung; RIVERS, Dean, Andrews
Patent: WO2012/170752 A1, 2012 ;
Location in patent: Page/Page column 58-59 ;
WO 2012/170752 A1