5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-7-甲苯磺酰-7h-吡咯并[2,3-d]嘧啶合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in ethylene glycol dimethyl ether
T=150°C; 0.166667 h; microwave irradiation;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED
Patent: WO2007/41130 A2, 2007 ;
Location in patent: Page/Page column 40-41; Sheet 1/9 ;
WO 2007/041130 A2